Novel pyrazole-containing compounds active against mycobacterium tuberculosis
2019-01-01 Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy
2021-01-01 Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis
2021-01-01 Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M.
COX inhibitors: a patent review (2011 - 2014)
2015-01-01 Consalvi, Sara; Biava, Mariangela; Poce, Giovanna
Anti-miRNA103/107 encapsulated in transferrin-conjugated lipid nanoparticles crosses blood-brain barrier and reduces brain ischemic damage
2024-01-01 Cepparulo, P.; Cuomo, O.; Campani, Virginia; Vinciguerra, A.; Sisalli, M. J.; Nele, V.; Anzilotti, S.; Valsecchi, V.; Casamassa, A.; Brancaccio, P.; Scorziello, A.; De Rosa, G.; Annunziato, L.; Pignataro., G.
Pharmaceutical salt of BM635 with improved bioavailability
2017-01-01 Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development?
2019-01-01 Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target
2016-01-01 Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction
2013-01-01 Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V.
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances
2023-01-01 Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects
2019-01-01 Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I
In vivo potent BM635 analogue with improved drug-like properties
2018-01-01 Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis
2016-01-01 Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents
2017-01-01 Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis
2020-01-01 Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G.
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors
2014-01-01 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors
2015-01-01 Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela
Overcoming drug resistance in TB: an update
2020-01-01 Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M.
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis
2021-01-01 Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G.
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme
2012-01-01 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Novel pyrazole-containing compounds active against mycobacterium tuberculosis | 1-gen-2019 | Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela | |
| Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy | 1-gen-2021 | Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria | |
| Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis | 1-gen-2021 | Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M. | |
| COX inhibitors: a patent review (2011 - 2014) | 1-gen-2015 | Consalvi, Sara; Biava, Mariangela; Poce, Giovanna | |
| Anti-miRNA103/107 encapsulated in transferrin-conjugated lipid nanoparticles crosses blood-brain barrier and reduces brain ischemic damage | 1-gen-2024 | Cepparulo, P.; Cuomo, O.; Campani, Virginia; Vinciguerra, A.; Sisalli, M. J.; Nele, V.; Anzilotti, S.; Valsecchi, V.; Casamassa, A.; Brancaccio, P.; Scorziello, A.; De Rosa, G.; Annunziato, L.; Pignataro., G. | |
| Pharmaceutical salt of BM635 with improved bioavailability | 1-gen-2017 | Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela | |
| Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development? | 1-gen-2019 | Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna | |
| MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target | 1-gen-2016 | Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
| The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction | 1-gen-2013 | Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V. | |
| Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances | 1-gen-2023 | Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna | |
| Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects | 1-gen-2019 | Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I | |
| In vivo potent BM635 analogue with improved drug-like properties | 1-gen-2018 | Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela | |
| A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis | 1-gen-2016 | Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela | |
| 1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents | 1-gen-2017 | Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
| Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis | 1-gen-2020 | Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G. | |
| Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors | 1-gen-2014 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini | |
| Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors | 1-gen-2015 | Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela | |
| Overcoming drug resistance in TB: an update | 1-gen-2020 | Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M. | |
| 6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis | 1-gen-2021 | Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G. | |
| Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme | 1-gen-2012 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini |
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